Masci, Domiziana
Masci, Domiziana
ROMA - Dipartimento di Scienze biotecnologiche di base, cliniche intensivologiche e perioperatorie
CHAPTER 4. Biocatalysis, an Introduction. Exploiting Enzymes as Green Catalysts in the Synthesis of Chemicals and Drugs
2021 Masci, Domiziana; Castagnolo, Daniele
Biocatalytic and Chemo-Enzymatic Approaches for the Synthesis of Heterocycles
2020 Zhao, F.; Masci, Domiziana; Tomarelli, E.; Castagnolo, D.
Monoamine Oxidase (MAO-N) Biocatalyzed Synthesis of Indoles from Indolines Prepared via Photocatalytic Cyclization/Arylative Dearomatization
2020 Zhao, F.; Masci, Domiziana; Ferla, S.; Varricchio, C.; Brancale, A.; Colonna, S.; Black, G. W.; Turner, N. J.; Castagnolo, D.
New indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains
2020 Nalli, M.; Armijos Rivera, J. I.; Masci, Domiziana; Coluccia, A.; Badia, R.; Riveira-Munoz, E.; Brambilla, Alberto; Cinquina, E.; Turriziani, O.; Falasca, F.; Catalano, M.; Limatola, Carlo; Este, J. A.; Maga, G.; Silvestri, R.; Crespan, E.; La Regina, Giuseppe
A facile and regioselective multicomponent synthesis of chiral aryl-1,2-mercaptoamines in water followed by monoamine oxidase (MAO-N) enzymatic resolution
2019 Lauder, K.; Masci, Domiziana; Toscani, A.; Al Mekdad, A.; Black, G. W.; Brown, N. L.; Turner, N. J.; Luisi, R.; Castagnolo, D.
Biocatalytic aromatization of indolines into indoles by monoamine oxidase (MAO-N) whole cells
2019 Masci, Domiziana; Zhao, F.; Colonna, S.; Black, G.; Turner, N. J.; Castagnolo, Daniele
Design, synthesis and biological evaluation of PDZ1 targeting NHERF1 inhibitors as anticancer agents
2019 La Regina, Giuseppe; Naccarato, V.; Masci, Domiziana; Puxeddu, M.; Bufano, Maria Oliva; Nalli, M.; Coluccia, A.; Orlando, Vittorio; Canettieri, G.; Gianni, Silvia Maria; Silvestri, R.
Small molecule inhibitors of kdm5 histone demethylases increase the radiosensitivity of breast cancer cells overexpressing JARID1B
2019 La Regina, Giuseppe; Naccarato, Valentina; Masci, Domiziana; Puxeddu, Michela; Nalli, Marianna; Coluccia, Antonio; Negri, Rodolfo; Silvestri, Romano
Switching on the activity of 1,5-diaryl-pyrrole derivatives against drug-resistant ESKAPE bacteria
2019 Masci, Domiziana; Sutton, Mark; Castagnolo, Daniele
Switching on the activity of 1,5-diaryl-pyrrole derivatives against drug-resistant ESKAPE bacteria: Structure-activity relationships and mode of action studies
2019 Masci, Domiziana; Hind, C.; Islam, M. K.; Toscani, A.; Clifford, M.; Coluccia, A.; Conforti, I.; Touitou, M.; Memdouh, S.; Wei, X.; La Regina, G.; Silvestri, R.; Sutton, J. M.; Castagnolo, D.
Indolylarylsulfones as novel potent anti-HIV-1 agents
2018 Masci, Domiziana; La Regina, Giuseppe; Coluccia, Antonio; Brancale, Andrea; Estè Josè, A.; Silvestri, Romano
Indolylarylsulfones as novel potent anti-HIV-1 agents
2018 Masci, Domiziana; La Regina, Giuseppe; Coluccia, Antonio; Andrea, Brancale; José A., Esté; Silvestri, Romano
New 6- and 7-heterocyclyl-1H-indole derivatives as potent tubulin assembly and cancer cell growth inhibitors
2018 La Regina, Giuseppe; Bai, R.; Coluccia, A.; Naccarato, V.; Famiglini, V.; Nalli, M.; Masci, Domiziana; Verrico, A.; Rovella, P.; Mazzoccoli, C.; Da Pozzo, E.; Cavallini, C.; Martini, Maria Cristina; Vultaggio, S.; Dondio, G.; Varasi, M.; Mercurio, C.; Hamel, E.; Lavia, P.; Silvestri, R.
Chiral Indolylarylsulfone Non-Nucleoside Reverse Transcriptase Inhibitors as New Potent and Broad Spectrum Anti-HIV-1 Agents
2017 Famiglini, V.; La Regina, G.; Coluccia, A.; Masci, D.; Brancale, A.; Badia, R.; Riveira-Munoz, E.; Este, J. A.; Crespan, E.; Brambilla, A.; Maga, G.; Catalano, M.; Limatola, C.; Formica, F. R.; Cirilli, R.; Novellino, E.; Silvestri, R.
Drug design and synthesis of new indolylarylsulfones as HIV-1 non-nucleoside reverse transcriptase inhibitors
2017 Famiglini, Valeria; La Regina, Giuseppe; Coluccia, Antonio; Masci, Domiziana; Roger, Badia; José A., Esté; Emmanuele, Crespan; Giovanni, Maga
Drug design and synthesis of new indolylarylsulfones as HIV-1 non-nucleoside reverse transcriptase inhibitors
2017 Masci, Domiziana; La Regina, Giuseppe; Famiglini, Valeria; Coluccia, Antonio; Brancale, Andrea; José A., Esté; Silvestri, Romano
Inhibition of dengue virus replication by novel inhibitors of RNA-dependent RNA polymerase and protease activities
2017 Pelliccia, S.; Wu, Y. -H.; Coluccia, A.; La Regina, Giuseppe; Tseng, C. -K.; Famiglini, V.; Masci, Domiziana; Hiscott, J.; Lee, J. -C.; Silvestri, R.
| Data di pubblicazione | Titolo | Autore(i) | File |
|---|---|---|---|
| 1-gen-2021 | CHAPTER 4. Biocatalysis, an Introduction. Exploiting Enzymes as Green Catalysts in the Synthesis of Chemicals and Drugs | Masci, Domiziana; Castagnolo, Daniele | |
| 1-gen-2020 | Biocatalytic and Chemo-Enzymatic Approaches for the Synthesis of Heterocycles | Zhao, F.; Masci, Domiziana; Tomarelli, E.; Castagnolo, D. | |
| 1-gen-2020 | Monoamine Oxidase (MAO-N) Biocatalyzed Synthesis of Indoles from Indolines Prepared via Photocatalytic Cyclization/Arylative Dearomatization | Zhao, F.; Masci, Domiziana; Ferla, S.; Varricchio, C.; Brancale, A.; Colonna, S.; Black, G. W.; Turner, N. J.; Castagnolo, D. | |
| 1-gen-2020 | New indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains | Nalli, M.; Armijos Rivera, J. I.; Masci, Domiziana; Coluccia, A.; Badia, R.; Riveira-Munoz, E.; Brambilla, Alberto; Cinquina, E.; Turriziani, O.; Falasca, F.; Catalano, M.; Limatola, Carlo; Este, J. A.; Maga, G.; Silvestri, R.; Crespan, E.; La Regina, Giuseppe | |
| 1-gen-2019 | A facile and regioselective multicomponent synthesis of chiral aryl-1,2-mercaptoamines in water followed by monoamine oxidase (MAO-N) enzymatic resolution | Lauder, K.; Masci, Domiziana; Toscani, A.; Al Mekdad, A.; Black, G. W.; Brown, N. L.; Turner, N. J.; Luisi, R.; Castagnolo, D. | |
| 1-gen-2019 | Biocatalytic aromatization of indolines into indoles by monoamine oxidase (MAO-N) whole cells | Masci, Domiziana; Zhao, F.; Colonna, S.; Black, G.; Turner, N. J.; Castagnolo, Daniele | |
| 1-gen-2019 | Design, synthesis and biological evaluation of PDZ1 targeting NHERF1 inhibitors as anticancer agents | La Regina, Giuseppe; Naccarato, V.; Masci, Domiziana; Puxeddu, M.; Bufano, Maria Oliva; Nalli, M.; Coluccia, A.; Orlando, Vittorio; Canettieri, G.; Gianni, Silvia Maria; Silvestri, R. | |
| 1-gen-2019 | Small molecule inhibitors of kdm5 histone demethylases increase the radiosensitivity of breast cancer cells overexpressing JARID1B | La Regina, Giuseppe; Naccarato, Valentina; Masci, Domiziana; Puxeddu, Michela; Nalli, Marianna; Coluccia, Antonio; Negri, Rodolfo; Silvestri, Romano | |
| 1-gen-2019 | Switching on the activity of 1,5-diaryl-pyrrole derivatives against drug-resistant ESKAPE bacteria | Masci, Domiziana; Sutton, Mark; Castagnolo, Daniele | |
| 1-gen-2019 | Switching on the activity of 1,5-diaryl-pyrrole derivatives against drug-resistant ESKAPE bacteria: Structure-activity relationships and mode of action studies | Masci, Domiziana; Hind, C.; Islam, M. K.; Toscani, A.; Clifford, M.; Coluccia, A.; Conforti, I.; Touitou, M.; Memdouh, S.; Wei, X.; La Regina, G.; Silvestri, R.; Sutton, J. M.; Castagnolo, D. | |
| 1-gen-2018 | Indolylarylsulfones as novel potent anti-HIV-1 agents | Masci, Domiziana; La Regina, Giuseppe; Coluccia, Antonio; Brancale, Andrea; Estè Josè, A.; Silvestri, Romano | |
| 1-gen-2018 | Indolylarylsulfones as novel potent anti-HIV-1 agents | Masci, Domiziana; La Regina, Giuseppe; Coluccia, Antonio; Andrea, Brancale; José A., Esté; Silvestri, Romano | |
| 1-gen-2018 | New 6- and 7-heterocyclyl-1H-indole derivatives as potent tubulin assembly and cancer cell growth inhibitors | La Regina, Giuseppe; Bai, R.; Coluccia, A.; Naccarato, V.; Famiglini, V.; Nalli, M.; Masci, Domiziana; Verrico, A.; Rovella, P.; Mazzoccoli, C.; Da Pozzo, E.; Cavallini, C.; Martini, Maria Cristina; Vultaggio, S.; Dondio, G.; Varasi, M.; Mercurio, C.; Hamel, E.; Lavia, P.; Silvestri, R. | |
| 1-gen-2017 | Chiral Indolylarylsulfone Non-Nucleoside Reverse Transcriptase Inhibitors as New Potent and Broad Spectrum Anti-HIV-1 Agents | Famiglini, V.; La Regina, G.; Coluccia, A.; Masci, D.; Brancale, A.; Badia, R.; Riveira-Munoz, E.; Este, J. A.; Crespan, E.; Brambilla, A.; Maga, G.; Catalano, M.; Limatola, C.; Formica, F. R.; Cirilli, R.; Novellino, E.; Silvestri, R. | |
| 1-gen-2017 | Drug design and synthesis of new indolylarylsulfones as HIV-1 non-nucleoside reverse transcriptase inhibitors | Famiglini, Valeria; La Regina, Giuseppe; Coluccia, Antonio; Masci, Domiziana; Roger, Badia; José A., Esté; Emmanuele, Crespan; Giovanni, Maga | |
| 1-gen-2017 | Drug design and synthesis of new indolylarylsulfones as HIV-1 non-nucleoside reverse transcriptase inhibitors | Masci, Domiziana; La Regina, Giuseppe; Famiglini, Valeria; Coluccia, Antonio; Brancale, Andrea; José A., Esté; Silvestri, Romano | |
| 1-gen-2017 | Inhibition of dengue virus replication by novel inhibitors of RNA-dependent RNA polymerase and protease activities | Pelliccia, S.; Wu, Y. -H.; Coluccia, A.; La Regina, Giuseppe; Tseng, C. -K.; Famiglini, V.; Masci, Domiziana; Hiscott, J.; Lee, J. -C.; Silvestri, R. |